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Antidepressant effects of 3‐‐2E‐propenoic acid isobutyl amide involve TSPO‐mediated mitophagy signalling pathway

  • 【作者】Qiang Wei,Wangyi Zhou,Ji Zheng,Dongmei Li,Mingyang Wang,Lu Feng,Wei Huang,Nan Yang,Min Han,Xiaohui Ma,Yanyong Liu
  • 【作者单位】Medical College, Tibet University, Lhasa, China;Pharmacology and Toxicology Research Centre, Tasly Institute, Tasly Holding Group Co., Ltd., Tianjin, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Pharmacology and Toxicology Research Centre, Tasly Institute, Tasly Holding Group Co., Ltd., Tianjin, China;Pharmacology and Toxicology Research Centre, Tasly Institute, Tasly Holding Group Co., Ltd., Tianjin, China;Yanyong Liu, Medical College, Tibet University, Tibet Autonomous Region, Lhasa, 850000, China;Department of Pharmacology, Institute of Basic Medical Sciences, Center of Neuroscience, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, 5 Dong Dan San Tiao, Beijing 100005, China.;Xiaohui Ma, Pharmacology and Toxicology Research Centre, Tasly Institute, Tasly Holding Group Co., Ltd., 2 East Pu Ji He Road, Beichen District, Tianjin 300410, China.;Medical College, Tibet University, Lhasa, China;Department of Pharmacology, Institute of Basic Medical Sciences, Neuroscience Center, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, Beijing, China;Yanyong Liu, Medical College, Tibet University, Tibet Autonomous Region, Lhasa, 850000, China;Department of Pharmacology, Institute of Basic Medical Sciences, Center of Neuroscience, Chinese Academy of Medical Sciences &School of Basic Medicine, Peking Union Medical College, 5 Dong Dan San Tiao, Beijing 100005, China.;Xiaohui Ma, Pharmacology and Toxicology Research Centre, Tasly Institute, Tasly Holding Group Co., Ltd., 2 East Pu Ji He Road, Beichen District, Tianjin 300410, China.
  • 【年份】2020
  • 【卷号】Vol.127 No.5
  • 【页码】380-388
  • 【ISSN】1742-7843
  • 【关键词】depression learned helplessness mitochondria mitophagy Piper laetispicum social defeat stress 
  • 【摘要】 Piper laetispicum C. DC is one of the Chinese herbal medicines used for alleviating depressive disorders. G11‐5 [3‐‐2E‐propenoic acid isobutyl amide] is synthesized based on the chemical structure of an active integrant of Piper laetispicum C. DC. Th...
  • 【文献类型】 期刊
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